5F-UR144、XLR-11 CAS 1364933-54-9

5F-UR144、XLR-11 CAS 1364933-54-9

撃た説明:

5F-UR144、XLR-11 CAS 1364933-54-9 XLR-11(5 " - フルオロ-UR-144)98 nmおよび83のEC50値とカンナビノイド受容体CB1とCB2のための強力なアゴニストとして作用する薬剤でありますnMで、respectively.Itは、UR-144、-796260およびA-834735のような化合物に関連する3-(tetramethylcyclopropylmethanoyl)インドール誘導体であるが、それは、具体的には、これらの他の類似の化合物と一緒に、特許や科学文献に記載されていない、と以前、アボット社がなされていないように見えます...

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説明:

5f-ur144-phoenixchem

5F-UR144,XLR-11 CAS 1364933-54-9

XLR-11 (5″-fluoro-UR-144) is a drug that acts as a potent agonist for the cannabinoid receptors CB1 and CB2 with EC50 values of 98 nM and 83 nM, respectively.It is a 3-(tetramethylcyclopropylmethanoyl)indole derivative related to compounds such as UR-144, A-796,260 and A-834,735, but it is not specifically listed in the patent or scientific literature alongside these other similar compounds,and appears to have not previously been made by Abbott Laboratories, despite falling within the claims of patent WO 2006/069196. XLR-11 was found to produce rapid, short-lived hypothermic effects in rats at doses of 3 mg/kg and 10 mg/kg, suggesting that it is of comparable potency to APICA and STS-135.

工厂5

5F-UR144,XLR-11


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