5F-UR144, XLR-11 CAS 1364933-54-9

5F-UR144, XLR-11 CAS 1364933-54-9

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5F-UR144, XLR-11 CAS 1364933-54-9 XLR-11 (5 "-fluoro-UR-144) adalah ubat yang bertindak sebagai agonis mujarab untuk reseptor cannabinoid CB1 dan CB2 dengan nilai EC50 98 nM dan 83 nM, respectively.It ialah 3- (tetramethylcyclopropylmethanoyl) indole terbitan yang berkaitan dengan sebatian seperti UR-144, a-796.260 dan a-834.735, tetapi ia tidak disenaraikan secara khusus dalam paten atau kesusasteraan saintifik di samping kewujudan sebatian lain yang serupa, dan nampaknya telah tidak telah dibuat oleh Abbott ...

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5f-ur144-phoenixchem

5F-UR144,XLR-11 CAS 1364933-54-9

XLR-11 (5″-fluoro-UR-144) is a drug that acts as a potent agonist for the cannabinoid receptors CB1 and CB2 with EC50 values of 98 nM and 83 nM, respectively.It is a 3-(tetramethylcyclopropylmethanoyl)indole derivative related to compounds such as UR-144, A-796,260 and A-834,735, but it is not specifically listed in the patent or scientific literature alongside these other similar compounds,and appears to have not previously been made by Abbott Laboratories, despite falling within the claims of patent WO 2006/069196. XLR-11 was found to produce rapid, short-lived hypothermic effects in rats at doses of 3 mg/kg and 10 mg/kg, suggesting that it is of comparable potency to APICA and STS-135.

工厂5

5F-UR144,XLR-11


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