5F-UR144,XLR-11 CAS 1364933-54-9

5F-UR144,XLR-11 CAS 1364933-54-9

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5F-UR144,XLR-11 CAS 1364933-54-9 XLR-11(5“ - 氟UR-144)是充当用于大麻素受体CB1和CB2与98纳米和83的EC 50值强效激动剂的药物纳米,respectively.It是与诸如UR-144,A-796260和A-834735的化合物3-(tetramethylcyclopropylmethanoyl)吲哚衍生物,但没有具体的专利或科学文献沿着这些其它类似化合物列出,并且似乎以前没有由Abbott制成...

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5f-ur144-phoenixchem

5F-UR144,XLR-11 CAS 1364933-54-9

XLR-11 (5″-fluoro-UR-144) is a drug that acts as a potent agonist for the cannabinoid receptors CB1 and CB2 with EC50 values of 98 nM and 83 nM, respectively.It is a 3-(tetramethylcyclopropylmethanoyl)indole derivative related to compounds such as UR-144, A-796,260 and A-834,735, but it is not specifically listed in the patent or scientific literature alongside these other similar compounds,and appears to have not previously been made by Abbott Laboratories, despite falling within the claims of patent WO 2006/069196. XLR-11 was found to produce rapid, short-lived hypothermic effects in rats at doses of 3 mg/kg and 10 mg/kg, suggesting that it is of comparable potency to APICA and STS-135.

工厂5

5F-UR144,XLR-11


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